SCHEMBL578265

SCHEMBL578265

O=C1C(=O)N(Cc2ccccc2)c2ccc(F)cc21

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARK7 Q99497 2/20 0.74
ALDH1A1 P00352 7/20 0.71
ALDH3A1 P30838 7/20 0.71
ALDH2 P05091 3/20 0.71
CHRM5 P08912 2/20 0.71
CHRM1 P11229 1/20 0.67
CES1 P23141 1/20 0.67
TRPA1 O75762 1/20 0.66
CA1 P00915 3/20 0.64
CA2 P00918 3/20 0.64
CA9 Q16790 3/20 0.64
CA12 O43570 2/20 0.64
CASP1 P29466 1/20 0.63
CASP3 P42574 1/20 0.63
CASP4 P49662 1/20 0.63
CASP7 P55210 1/20 0.63
CASP9 P55211 1/20 0.63
CASP6 P55212 1/20 0.63
CASP8 Q14790 1/20 0.63
NSD2 O96028 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12930212 0.88 ALDH1A1 (0.67) PARK7ALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL4597660 0.87 CHRM5 (0.73) PARK7ALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL10369984 0.84 CHRM5 (0.58) PARK7ALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL9097463 0.83 PARK7 (0.67) PARK7ALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL16798714 0.83 ALDH3A1 (1.00) ALDH1A1ALDH3A1ALDH2CHRM1CES1
SCHEMBL10979016 0.83 ALDH1A1 (0.69) PARK7ALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL30937981 0.83 CHRM5 (1.00) PARK7ALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL28365954 0.82 TRPA1 (0.59) PARK7ALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL3021031 0.82 CHRM5 (0.72) PARK7ALDH1A1ALDH3A1CHRM5CA1
SCHEMBL13627936 0.82 TRPA1 (0.62) PARK7ALDH1A1ALDH3A1ALDH2CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118459390-B 3-Hydroxy oxindole derivative containing Z-type 1, 4-dicarbonyl olefin, and preparation method and application thereof SUN YAT-SEN UNIVERSITY (CN) 2026-05-26 CN disclosed
EP-4536642-A1 HETEROCYCLIC COMPOUNDS AS PI3KA INHIBITORS Synnovation Therapeutics, Inc. (US) 2025-04-16 EP disclosed
CN-118459390-A 3-Hydroxy oxindole derivative containing Z-type 1, 4-dicarbonyl olefin, and preparation method and application thereof 中山大学 2024-08-09 CN disclosed
WO-2023239846-A1 HETEROCYCLIC COMPOUNDS AS PI3KΑ INHIBITORS SYNNOVATION THERAPEUTICS, INC. (US) 2023-12-14 WO disclosed
WO-2023239846-A1 HETEROCYCLIC COMPOUNDS AS PI3KΑ INHIBITORS SYNNOVATION THERAPEUTICS, INC. (US) 2023-12-14 WO disclosed
CN-112920191-B Arylethynyl oxindole oxirane as well as preparation method and application thereof 南宁师范大学 2022-03-25 CN disclosed
US-RE47731-E1 Kinase inhibitors and method of treating cancer with same UNIV HEALTH NETWORK (CA) 2019-11-19 US disclosed
US-10358436-B2 Kinase inhibitors and method of treating cancer UNIVERSITY HEALTH NETWORK (CA) 2019-07-23 US disclosed
US-20180282306-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER UNIVERSITY HEALTH NETWORK (CA) 2018-10-04 US disclosed
US-10077255-B2 Synthesis of chiral 2-(1H-indazol-6-yl)-spiro[cyclopropane-1,3′-indolin]-2′-ones UNIVERSITY HEALTH NETWORK (CA) 2018-09-18 US disclosed
US-20120149686-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORKS (CA) 2012-06-14 US disclosed
EP-2417127-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME University Health Network (CA) 2012-02-15 EP disclosed
US-20110263598-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER UNIVERSITY HEALTH NETWORKS (CA) 2011-10-27 US disclosed
WO-2011123946-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed
WO-2011123947-A1 SYNTHESIS OF CHIRAL 2-(1H-INDAZOL-6-YL)-SPIRO[CYCLOPROPANE-1,3'- INDOLIN]-2'-ONES UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed
US-20110009379-A1 INDOLINONE COMPOUND ASTELLAS PHARMA INC. (JP) 2011-01-13 US disclosed
US-20110009379-A1 INDOLINONE COMPOUND ASTELLAS PHARMA INC. (JP) 2011-01-13 US disclosed
EP-2261206-A1 INDOLINONE COMPOUND Astellas Pharma Inc. (JP) 2010-12-15 EP disclosed
WO-2010115279-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2010-10-14 WO disclosed
WO-2009123080-A1 INDOLINONE COMPOUND アステラス製薬株式会社 (JP) 2009-10-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149686-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME MAP3K5, MAP3K6, MAP3K1 PARK7 3331/4885ALDH1A1 2633/4885ALDH3A1 2473/4885
US-20110263598-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER MAP3K6, MAP3K5, MAP3K19 PARK7 3683/4885ALDH1A1 2389/4885ALDH3A1 2333/4885
US-10358436-B2 Kinase inhibitors and method of treating cancer MAP3K6, MAP3K5, MAP3K19 PARK7 3683/4885ALDH1A1 2389/4885ALDH3A1 2333/4885
US-20110009379-A1 INDOLINONE COMPOUND TRPA1, TRPV1, TRPV6 PARK7 516/4885ALDH1A1 1687/4885ALDH3A1 2467/4885
US-10077255-B2 Synthesis of chiral 2-(1H-indazol-6-yl)-spiro[cyclopropane-1,3′-indolin]-2′-ones IDO1, IDO2, IMPA1 PARK7 902/4885ALDH1A1 238/4885ALDH3A1 263/4885
US-20180282306-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER MAP3K6, MAP3K5, MAP3K19 PARK7 3683/4885ALDH1A1 2389/4885ALDH3A1 2333/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.