SCHEMBL5789256

SCHEMBL5789256

COc1ccc[c]c1-c1ccc(S(C)(=O)=O)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.46
SMN1; SMN2 Q16637 1/20 0.43
KMT2A Q03164 1/20 0.41
PTGDR2 Q9Y5Y4 2/20 0.41
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
CCNT1 O60563 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK9 P50750 1/20 0.38
PTGS1 P23219 2/20 0.37
STK10 O94804 1/20 0.37
SLK Q9H2G2 1/20 0.37
LRRK2 Q5S007 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512743 0.77 PTGS2 (0.46) PTGS2SMN1; SMN2PTGS1
SCHEMBL4284342 0.75 HTR7 (0.40) SMN1; SMN2KMT2A
SCHEMBL28986621 0.73 PTGS2 (0.41) PTGS2KMT2APTGDR2CYP11B1CYP11B2
SCHEMBL27732214 0.72 PTGS2 (0.57) PTGS2SMN1; SMN2PTGS1
SCHEMBL4637513 0.70 PTGS2 (0.43) PTGS2SMN1; SMN2PTGDR2CYP11B1CYP11B2
SCHEMBL13211354 0.70 ALDH1A1 (0.63) PTGS2SMN1; SMN2KMT2A
SCHEMBL2885322 0.69 CA1 (0.50) SMN1; SMN2PTGS1
SCHEMBL6402326 0.68 PTGS2 (0.52) PTGS2SMN1; SMN2KMT2APTGS1
SCHEMBL2372578 0.68 APP (0.47) PTGS2SMN1; SMN2KMT2APTGS1
SCHEMBL11523591 0.68 CYP1A1 (0.53) SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660500-A1 SUBSTITUTED IMIDAZOPYRIMIDINES FOR THE PREVENTION AND TREATMENT OF CANCER LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2006-05-31 EP disclosed
WO-2005014598-A1 SUBSTITUTED IMIDAZOPYRIMIDINES FOR THE PREVENTION AND TREATMENT OF CANCER LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2005-02-17 WO disclosed