SCHEMBL5791966

SCHEMBL5791966

COc1cccc(C(=O)NN(CC(C)(C)C)c2ccnc(C#N)n2)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.45
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
ABCB1 P08183 1/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
GRM5 P41594 1/20 0.40
FGFR4 P22455 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 3/20 0.39
TP53 P04637 2/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5792274 0.90 CTSK (0.43) CTSKCTSS
SCHEMBL8268811 0.86 TAS1R3 (0.40) CTSKCTSLCTSSNPC1RAB9A
SCHEMBL8270702 0.86 NPC1 (0.46) CTSKCTSLCTSSNPC1RAB9A
Trifluoroacetic Acid SCHEMBL5794693 0.83 TSHR (0.38) CTSKCTSLCTSSABCB1NPC1
SCHEMBL5790636 0.82 CTSK (0.44) CTSKCTSLCTSSFGFR4
SCHEMBL8268817 0.80 CTSK (0.43) CTSKCTSLCTSSNPC1RAB9A
SCHEMBL5793789 0.79 LMNA (0.43) CTSKCTSLCTSSNPC1RAB9A
SCHEMBL5793805 0.77 CTSK (0.52) CTSKCTSLCTSSFGFR4
SCHEMBL5790947 0.77 MCHR1 (0.52) CTSKNPC1RAB9AMEN1KMT2A
SCHEMBL8269394 0.75 CTSL (0.45) CTSKCTSLCTSSNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed