SCHEMBL5790959

SCHEMBL5790959

NC(=O)N1CCNCC1(c1ccccc1)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.35
HTR2A P28223 3/20 0.34
OPRD1 P41143 1/20 0.34
PDK2 Q15119 1/20 0.34
TACR1 P25103 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TSHR P16473 2/20 0.33
OPRM1 P35372 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
POLB P06746 2/20 0.32
USP2 O75604 1/20 0.32
HSD17B10 Q99714 1/20 0.32
RORC P51449 1/20 0.32
CYP2D6 P10635 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
MLYCD O95822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29761590 0.89 SIGMAR1 (0.36) SIGMAR1HTR2AOPRD1PDK2TACR1
SCHEMBL2404059 0.86 SIGMAR1 (0.35) SIGMAR1HTR2AOPRD1PDK2TACR1
SCHEMBL30479863 0.82 VNN1 (0.33)
SCHEMBL5792213 0.81 HSD11B1 (0.37) OPRD1OPRM1TDP1MLYCDCHRM2
SCHEMBL25424435 0.80 EPHX2 (0.33) ALDH1A1KDM4E
SCHEMBL5790641 0.79 HSD11B1 (0.39) ALDH1A1TSHROPRM1KDM4EMAPT
SCHEMBL17372634 0.78 OPRM1 (0.33) SIGMAR1HTR2AOPRD1TACR1OPRM1
SCHEMBL5822059 0.78 MEN1 (0.42) SIGMAR1OPRD1ALDH1A1TSHROPRM1
SCHEMBL4592731 0.77 SIGMAR1 (0.38) SIGMAR1HTR2AOPRD1ALDH1A1TSHR
SCHEMBL4759637 0.76 HTR2A (0.38) SIGMAR1HTR2AOPRD1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1483241-A4 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2006-12-13 EP claimed
EP-1483241-A2 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Company (US) 2004-12-08 EP claimed
WO-2003075853-A2 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2003-09-18 WO claimed