SCHEMBL5791389

SCHEMBL5791389

CC(C)CN(NC(=O)c1ccccc1)c1ccnc(C#N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 7/20 0.46
CTSB P07858 6/20 0.46
CTSK P43235 5/20 0.46
CTSS P25774 5/20 0.46
FGFR4 P22455 1/20 0.38
MAPK14 Q16539 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 2/20 0.35
POLB P06746 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
CTSF Q9UBX1 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
S1PR2 O95136 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8270696 0.89 CTSL (0.47) CTSLCTSBCTSKCTSSFGFR4
SCHEMBL8268809 0.88 CTSL (0.42) CTSLCTSBCTSKCTSSFGFR4
SCHEMBL8269394 0.87 CTSL (0.45) CTSLCTSBCTSKCTSSFGFR4
SCHEMBL8269396 0.87 CTSK (0.45) CTSLCTSBCTSKCTSSFGFR4
SCHEMBL8268811 0.87 TAS1R3 (0.40) CTSLCTSBCTSKCTSSFGFR4
Trifluoroacetic Acid SCHEMBL5794344 0.86 CTSL (0.43) CTSLCTSBCTSKCTSSFGFR4
Trifluoroacetic Acid SCHEMBL5794600 0.85 CTSL (0.41) CTSLCTSBCTSKCTSSFGFR4
SCHEMBL8270505 0.85 CTSK (0.42) CTSLCTSBCTSKCTSSFGFR4
SCHEMBL8271456 0.85 CTSK (0.47) CTSLCTSBCTSKCTSSFGFR4
SCHEMBL5793933 0.84 CTSK (0.39) CTSLCTSBCTSKCTSSFGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed