SCHEMBL8268809

SCHEMBL8268809

CC(C)CN(NC(=O)c1cccc(F)c1)c1ccnc(C#N)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.42
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.37
RAB9A P51151 2/20 0.37
ALDH1A1 P00352 1/20 0.37
FGFR4 P22455 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
NPC1 O15118 1/20 0.36
GPR139 Q6DWJ6 1/20 0.36
AR P10275 1/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
PKM P14618 1/20 0.35
MAPK1 P28482 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5794600 0.95 CTSL (0.41) CTSLCTSBCTSSCTSKMEN1
SCHEMBL8270696 0.88 CTSL (0.47) CTSLCTSBCTSSCTSKKMT2A
SCHEMBL5791389 0.88 CTSL (0.46) CTSLCTSBCTSSCTSKMEN1
SCHEMBL8268811 0.87 TAS1R3 (0.40) CTSLCTSBCTSSCTSKMEN1
SCHEMBL8271448 0.86 CTSK (0.46) CTSLCTSKMEN1KMT2ARAB9A
SCHEMBL8269989 0.85 NPC1 (0.44) MEN1KMT2ALMNARAB9AALDH1A1
SCHEMBL8270727 0.85 ANO1 (0.39) CTSLCTSBCTSSCTSKMEN1
Trifluoroacetic Acid SCHEMBL5794693 0.84 TSHR (0.38) CTSLCTSBCTSSCTSKMEN1
Trifluoroacetic Acid SCHEMBL5794344 0.83 CTSL (0.43) CTSLCTSBCTSSCTSKALDH1A1
SCHEMBL8269396 0.82 CTSK (0.45) CTSLCTSBCTSSCTSKLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed