SCHEMBL8269396

SCHEMBL8269396

CC(C)CN(NC(=O)c1ccc(C(F)(F)F)cc1)c1ccnc(C#N)n1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.45
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
CTSS P25774 1/20 0.45
TRPM8 Q7Z2W7 1/20 0.37
FGFR4 P22455 1/20 0.35
MMP3 P08254 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
VNN1 O95497 1/20 0.35
PDE2A O00408 1/20 0.35
TRPV3 Q8NET8 3/20 0.35
LMNA P02545 1/20 0.35
IDO1 P14902 1/20 0.35
TLR7 Q9NYK1 1/20 0.34
MLYCD O95822 1/20 0.34
HDAC4 P56524 2/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5794344 0.88 CTSL (0.43) CTSKCTSLCTSBCTSSFGFR4
SCHEMBL5791389 0.87 CTSL (0.46) CTSKCTSLCTSBCTSSFGFR4
SCHEMBL5794599 0.87 CTSK (0.38) CTSKCTSLCTSBCTSSMMP3
SCHEMBL8269394 0.86 CTSL (0.45) CTSKCTSLCTSBCTSSFGFR4
Trifluoroacetic Acid SCHEMBL5791067 0.85 CTSL (0.41) CTSKCTSLCTSBCTSSTRPM8
Trifluoroacetic Acid SCHEMBL5791991 0.84 FPR2 (0.40) IDO1
SCHEMBL8268809 0.82 CTSL (0.42) CTSKCTSLCTSBCTSSFGFR4
SCHEMBL8268851 0.82 CTSL (0.42) CTSKCTSLCTSBCTSSFGFR4
SCHEMBL5791497 0.81 CTSK (0.42) CTSKCTSLCTSBCTSSFGFR4
Trifluoroacetic Acid SCHEMBL5793410 0.80 CTSK (0.65) CTSKCTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed