SCHEMBL5798780

SCHEMBL5798780

CCCCCCCn1ccc2cc(-c3c(CC)cccc3CC)nc(C#N)c21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 12/20 0.38
GRM2 Q14416 1/20 0.33
CNR2 P34972 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
GLO1 Q04760 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
OXER1 Q8TDS5 1/20 0.31
ICMT O60725 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1762786 0.78 C5AR1 (0.31)
SCHEMBL5796068 0.75 TLR8 (0.40) TLR8GLO1KDM4ENPC1ALDH1A1
SCHEMBL5798513 0.65 CDK4 (0.38) TLR8CNR2ICMT
SCHEMBL2476855 0.64 GRM2 (0.38) GRM2CNR2SMN1; SMN2
SCHEMBL17304280 0.62 LNPEP (0.46) TLR8GRM2GLO1KDM4EALDH1A1
SCHEMBL17023237 0.62 LMNA (0.45) GRM2ALDH1A1SMN1; SMN2
SCHEMBL1328172 0.62 C5AR1 (0.46)
SCHEMBL201520 0.62 ACACB (0.45) GRM2CNR2ALDH1A1HPGDICMT
SCHEMBL28990232 0.61 BACE1 (0.46) GRM2CNR2OXER1
SCHEMBL28990233 0.61 OXER1 (0.46) TLR8CNR2OXER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006042102-A2 PYRROLO-PYRIDINE, PYRROLO-PYRIMIDINE AND RELATED HETEROCYCLIC COMPOUNDS NEUROGEN CORPORATION (US) 2006-04-20 WO disclosed