SCHEMBL5799447

SCHEMBL5799447

O=C(NO)c1ccc(C=C(CNc2ccc(-c3ccccc3)cc2)CC(O)c2cccc3ccccc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 13/20 0.43
HDAC8 Q9BY41 5/20 0.43
HDAC1 Q13547 13/20 0.40
HDAC3 O15379 4/20 0.40
HDAC4 P56524 4/20 0.40
HDAC7 Q8WUI4 4/20 0.40
HDAC2 Q92769 4/20 0.40
HDAC9 Q9UKV0 4/20 0.40
HDAC5 Q9UQL6 4/20 0.40
HDAC10 Q969S8 3/20 0.40
HDAC11 Q96DB2 3/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
P2RX3 P56373 1/20 0.39
PARP1 P09874 1/20 0.39
ACP3 P15309 1/20 0.38
APP P05067 1/20 0.36
ACHE P22303 1/20 0.36
NCOR2 Q9Y618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5797676 0.94 HDAC6 (0.42) HDAC6HDAC8HDAC1HDAC3HDAC4
SCHEMBL5796765 0.91 MAPT (0.41) ALDH1A1HPGDSMN1; SMN2ACP3
SCHEMBL5797642 0.89 HDAC6 (0.44) HDAC6HDAC8HDAC1HDAC3HDAC4
SCHEMBL5796436 0.83 HDAC1 (0.45) HDAC6HDAC8HDAC1HDAC3HDAC4
SCHEMBL5823657 0.82 ALDH1A1 (0.46) ALDH1A1HPGDSMN1; SMN2
SCHEMBL5797675 0.81 HDAC6 (0.42) HDAC6HDAC8HDAC1HDAC3HDAC4
SCHEMBL13850455 0.81 P2RX3 (0.58) HDAC6HDAC8HDAC1HDAC3HDAC4
SCHEMBL5799640 0.81 MAPT (0.52) ALDH1A1ACP3
SCHEMBL5799923 0.80 GCGR (0.43) ALDH1A1HPGD
SCHEMBL5796337 0.80 HDAC6 (0.38) HDAC6HDAC8HDAC1HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006025683-A1 ARYLAMINOMETHYL PROPENYL BENZHYDROXYAMID DERIVATIVES WITH INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-03-09 WO disclosed