SCHEMBL5799659

SCHEMBL5799659

COc1cccc(NCC(=Cc2ccc(C(=O)O)cc2)CC(O)c2cccc3ccccc23)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.41
MAPT P10636 5/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
NPC1 O15118 5/20 0.39
RAB9A P51151 5/20 0.39
CDC25B P30305 1/20 0.39
MITF O75030 1/20 0.39
ROCK2 O75116 1/20 0.38
GRK2 P25098 1/20 0.38
GRK5 P34947 1/20 0.38
GRK3 P35626 1/20 0.38
GAA P10253 2/20 0.38
GFER P55789 1/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5796946 0.93 MTNR1A (0.43) MTNR1AMAPTMEN1KMT2AALDH1A1
SCHEMBL5799923 0.91 GCGR (0.43) MTNR1AMAPTMEN1KMT2AKDM4E
SCHEMBL5799640 0.88 MAPT (0.52) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL5799682 0.85 NPC1 (0.39) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL5823657 0.85 ALDH1A1 (0.46) MTNR1AMAPTMEN1KMT2AALDH1A1
SCHEMBL5796765 0.83 MAPT (0.41) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL5822231 0.83 KMT2A (0.48) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL5799741 0.82 ALDH1A1 (0.40) MAPTKMT2AKDM4EALDH1A1NPC1
SCHEMBL5797676 0.80 HDAC6 (0.42) MAPTCYP2C9CYP2C19MCL1
SCHEMBL5797642 0.79 HDAC6 (0.44) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006025683-A1 ARYLAMINOMETHYL PROPENYL BENZHYDROXYAMID DERIVATIVES WITH INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-03-09 WO disclosed