SCHEMBL5799770

SCHEMBL5799770

CC(NC(=O)N1CCC2(CC1)C(=O)N(Cc1ccccc1)CN2c1ccccc1)C(NC(=O)C1C2CC3CC(C2)CC1C3)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.41
OPRK1 P41145 6/20 0.41
OPRL1 P41146 6/20 0.41
OPRD1 P41143 5/20 0.41
ENPP2 Q13822 3/20 0.41
BDKRB2 P30411 1/20 0.40
NPC1L1 Q9UHC9 1/20 0.39
DDR1 Q08345 1/20 0.39
MEN1 O00255 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP2C9 P11712 1/20 0.38
CCR3 P51677 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5780785 0.85 OPRM1 (0.41) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL6475235 0.83 OPRL1 (0.41) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL5802411 0.82 ENPP2 (0.46) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL5800911 0.82 NPC1L1 (0.49) OPRM1OPRK1OPRL1OPRD1NPC1L1
SCHEMBL5799004 0.81 ENPP2 (0.50) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL5802331 0.81 BDKRB2 (0.47) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL5799989 0.80 ENPP2 (0.44) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL5799178 0.79 ENPP2 (0.43) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL5783032 0.79 NPC1L1 (0.44) OPRM1OPRK1OPRL1OPRD1ENPP2
SCHEMBL5783117 0.78 OPRM1 (0.47) OPRM1OPRK1OPRL1OPRD1ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329451-B1 SPIRO COMPOUNDS AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES (JP) 2006-08-23 EP disclosed
EP-1329451-A1 SPIRO COMPOUNDS AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2003-07-23 EP disclosed