SCHEMBL5801705

SCHEMBL5801705

CCN(CC)C(=O)Cn1cc(C2CCN(C(=O)C3CCCC3)C2)c2ccccc21.Cn1cc(C2CCN(C=CC(=O)c3ccccc3)C2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.47
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 5/20 0.38
MEN1 O00255 3/20 0.37
MAPT P10636 2/20 0.37
IDE P14735 1/20 0.37
HRH2 P25021 3/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4859493 0.85 ALDH1A1 (0.50) RORCALDH1A1KMT2AMEN1MAPT
SCHEMBL4858049 0.81 MEN1 (0.52) RORCALDH1A1KMT2AMEN1MAPT
SCHEMBL5202233 0.74 HRH2 (0.41) ALDH1A1KMT2AMEN1MAPTHRH2
SCHEMBL5203151 0.73 ALDH1A1 (0.50) ALDH1A1KMT2AMEN1MAPTIDE
SCHEMBL4857600 0.68 HTR2A (0.49) ALDH1A1MAPTHRH2HTR2AHTR2C
SCHEMBL4849753 0.68 HRH2 (0.52) HRH2HTR2AHTR2CHTR2B
SCHEMBL5705162 0.66 RORC (0.51) RORCALDH1A1KMT2AMEN1CYP2C9
SCHEMBL4858050 0.66 RAB9A (0.62) RORCALDH1A1KMT2AMEN1MAPT
SCHEMBL4855807 0.65 KDM4E (0.48) RORCALDH1A1USP2
SCHEMBL5202270 0.65 MAPT (0.43) ALDH1A1KMT2AMEN1MAPTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2006-05-10 EP disclosed
WO-2005019208-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2005-03-03 WO disclosed