SCHEMBL5202233

SCHEMBL5202233

C#CCn1cc(C2CCN(C=CC(=O)c3ccccc3)C2)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 11/20 0.41
MAPT P10636 4/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
KMT2A Q03164 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TP53 P04637 1/20 0.38
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4858049 0.81 MEN1 (0.52) MAPTNPC1POLBHPGDNFKB1
SCHEMBL4857600 0.78 HTR2A (0.49) HRH2MAPTPOLBHTR2AHTR2C
SCHEMBL5206944 0.78 RAB9A (0.55) MAPTNPC1POLBHPGDRAB9A
SCHEMBL5801705 0.74 RORC (0.47) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL4849753 0.73 HRH2 (0.52) HRH2HTR2AHTR2CHTR2B
SCHEMBL5205671 0.69 MAPT (0.47) HRH2MAPTNPC1POLBHPGD
SCHEMBL5203557 0.69 ALDH1A1 (0.50) HRH2RAB9AKMT2AMEN1ALDH1A1
SCHEMBL6779805 0.68 HRH2 (0.75) HRH2HTR2AHTR2CHTR2B
SCHEMBL4859737 0.67 KMT2A (0.46) MAPTPOLBRAB9AKMT2AMEN1
SCHEMBL5201910 0.62 NPC1 (0.42) HRH2MAPTNPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed