SCHEMBL5809497

SCHEMBL5809497

Fc1cccc(-n2cnnn2)c1F

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
NPSR1 Q6W5P4 1/20 0.50
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 1/20 0.46
NOTUM Q6P988 4/20 0.46
RXRA P19793 3/20 0.41
GRIN1 Q05586 3/20 0.41
GRIN2B Q13224 3/20 0.41
PKM P14618 1/20 0.40
F2 P00734 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14242848 0.85 ALDH1A1 (0.58) ALDH1A1NPSR1KMT2AKDM4ENOTUM
SCHEMBL12615992 0.78 ALDH1A1 (0.68) ALDH1A1NPSR1KMT2AKDM4ENOTUM
SCHEMBL24427485 0.75 NOTUM (0.45) ALDH1A1NPSR1KMT2AKDM4ENOTUM
SCHEMBL30538055 0.74 KEAP1 (0.50) NOTUMRXRAGRIN1GRIN2B
SCHEMBL23118864 0.73 NOTUM (0.40) ALDH1A1NPSR1KMT2AKDM4ENOTUM
SCHEMBL28544293 0.71 MAPT (0.44) ALDH1A1NPSR1KMT2AKDM4ENOTUM
SCHEMBL30538087 0.71 RXRA (0.40) NOTUMRXRAGRIN1GRIN2B
SCHEMBL11146019 0.70 ALDH1A1 (0.54) ALDH1A1NPSR1KMT2AKDM4ENOTUM
SCHEMBL18378771 0.70 ALDH1A1 (0.54) ALDH1A1NPSR1KMT2AKDM4ENOTUM
SCHEMBL15879736 0.70 ALDH1A1 (1.00) ALDH1A1NPSR1KMT2AKDM4ENOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006086229-A1 THE USE OF SELECTIVE P2X7 RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2006-08-17 WO claimed