SCHEMBL5810901

SCHEMBL5810901

O=c1ccc(-c2c(-c3ccccc3)nn3cccnc23)n[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
PDE3A Q14432 6/20 0.46
PDE5A O76074 1/20 0.46
PDE3B Q13370 5/20 0.43
PTGS2 P35354 1/20 0.43
KCNQ3 O43525 2/20 0.38
KCNQ2 O43526 2/20 0.38
IGF1R P08069 2/20 0.37
MAPK3 P27361 1/20 0.36
MAPK1 P28482 1/20 0.36
MAPK14 Q16539 1/20 0.36
HPGD P15428 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
GPR119 Q8TDV5 1/20 0.36
ADORA1 P30542 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5810385 0.81 PDE3A (0.65) CYP1A2PDE3APDE5AIGF1RMAPK3
SCHEMBL17736144 0.78 PTGS2 (0.58) PDE3APDE3BPTGS2KCNQ3KCNQ2
SCHEMBL7369957 0.77 PDE3A (0.48) CYP1A2PDE3APDE5APDE3BIGF1R
SCHEMBL6824334 0.74 PDE3A (0.46) CYP1A2PDE3APDE5APDE3BPTGS2
SCHEMBL8888651 0.73 CYP1A2 (0.55) CYP1A2PDE3APDE5AMAPK1HPGD
SCHEMBL5946755 0.72 PTGS2 (0.42) PDE3APDE3BPTGS2KCNQ3KCNQ2
SCHEMBL5946616 0.72 HPGDS (0.43) PDE3APDE3BPTGS2KCNQ3KCNQ2
SCHEMBL6818685 0.71 PDE3A (0.47) CYP1A2PDE3APDE5AIGF1RMAPK3
SCHEMBL6539289 0.71 CYP1A2 (0.60) CYP1A2PDE3APDE3BPTGS2HPGD
SCHEMBL8836696 0.70 PTGS2 (0.62) PTGS2KCNQ3KCNQ2MAPK14JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006038734-A1 PYRIDAZINONE DERIVATIVES CYTOKINES INHIBITORS ASTELLAS PHARMA INC. (JP) 2006-04-13 WO disclosed