SCHEMBL5817545

SCHEMBL5817545

CNC(=N)c1c(SC)nc(-c2ccc(SC)cc2)n(-c2ccc(C(C)C)cc2)c1=O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
DHFR P00374 1/20 0.34
ESR1 P03372 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 2/20 0.31
UCHL3 P15374 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HTT P42858 1/20 0.31
HSP90AA1 P07900 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821043 0.90 ESR1 (0.35) ESR1ALDH1A1SMN1; SMN2HTTMAPT
SCHEMBL5821476 0.90 ALDH1A1 (0.43) ESR1ALDH1A1RXFP1SMN1; SMN2HTT
SCHEMBL5817584 0.88 PTGS2 (0.39) DHFRALDH1A1KMT2A
SCHEMBL5819664 0.86 PTGS2 (0.39) ESR1ALDH1A1CYP1A2CYP2C19
SCHEMBL5818149 0.85 ESR1 (0.34) TDP1ESR1ALDH1A1KMT2AMEN1
SCHEMBL5817548 0.82 DHFR (0.36) TDP1DHFRESR1ALDH1A1KMT2A
SCHEMBL5821416 0.81 AOC3 (0.42) ALDH1A1KMT2ACYP2C9CYP2C19SMN1; SMN2
SCHEMBL5817609 0.78 MAPK13 (0.39) ESR1ALDH1A1KMT2AMEN1RXFP1
SCHEMBL5821095 0.77 CA9 (0.43) ALDH1A1
SCHEMBL4853028 0.77 KDM4E (0.50) TDP1DHFRALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO claimed
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed