SCHEMBL5817609

SCHEMBL5817609

CNC(=N)c1c(SC)nc(-c2ccncc2)n(-c2ccc(F)cc2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 4/20 0.39
MAPK12 P53778 4/20 0.39
MAPK11 Q15759 4/20 0.39
MAPK14 Q16539 4/20 0.39
GCGR P47871 2/20 0.39
ALDH1A1 P00352 4/20 0.36
AOC3 Q16853 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GRIA1 P42261 1/20 0.34
CACNG8 Q8WXS5 1/20 0.34
CACNG2 Q9Y698 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HSD17B10 Q99714 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821416 0.89 AOC3 (0.42) ALDH1A1AOC3L3MBTL1KMT2A
SCHEMBL5820968 0.86 CA2 (0.38) KMT2A
SCHEMBL5821417 0.84 ALDH1A1 (0.36) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL5817785 0.84 ALDH1A1 (0.31) ALDH1A1ESR1
SCHEMBL5821476 0.82 ALDH1A1 (0.43) ALDH1A1NPSR1RXFP1LMNAESR1
SCHEMBL5817617 0.81 MAPK14 (0.36) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL5819664 0.81 PTGS2 (0.39) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL5821043 0.80 ESR1 (0.35) ALDH1A1AOC3ESR1
SCHEMBL5817545 0.78 TDP1 (0.36) ALDH1A1RXFP1MEN1KMT2AESR1
SCHEMBL5821095 0.78 CA9 (0.43) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed