SCHEMBL5819680

SCHEMBL5819680

Cc1c(C(C)C(=O)OC2CCCC2)c2c(F)c(O)ccc2n1C(=O)c1ccc(Cl)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.37
CYP19A1 P11511 1/20 0.33
PDE2A O00408 1/20 0.32
TACR3 P29371 5/20 0.31
TACR2 P21452 3/20 0.31
TACR1 P25103 2/20 0.31
KCNH2 Q12809 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
FAAH O00519 1/20 0.31
MGLL Q99685 1/20 0.31
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
TSHR P16473 1/20 0.30
USP14 P54578 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5822674 0.98 PTGS2 (0.36) PTGS2CYP19A1PDE2ATACR3TACR2
SCHEMBL5800554 0.94 PTGS2 (0.38) PTGS2CYP19A1AKR1C3AKR1C2TSHR
SCHEMBL5800295 0.92 TSHR (0.36) PTGS2CYP19A1AKR1C3AKR1C2TSHR
SCHEMBL5560260 0.92 PTGS2 (0.37) PTGS2CYP19A1FAAHMGLL
SCHEMBL5558388 0.91 PTGS2 (0.35) PTGS2CYP19A1AKR1C3AKR1C2FAAH
SCHEMBL5798701 0.90 PTGS2 (0.45) PTGS2CYP19A1AKR1C3AKR1C2
SCHEMBL5822558 0.89 PTGS2 (0.34) PTGS2CYP19A1PDE2ATACR3TACR2
SCHEMBL5800993 0.88 PTGS2 (0.37) PTGS2CYP19A1
SCHEMBL5559333 0.88 PTGS2 (0.43) PTGS2AKR1C3AKR1C2
SCHEMBL5819926 0.86 L3MBTL1 (0.37) PTGS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed