SCHEMBL5800295

SCHEMBL5800295

Cc1c(C(C)C(=O)OC2CCC2)c2c(F)c(O)ccc2n1C(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
PTGS2 P35354 1/20 0.36
HSD11B1 P28845 1/20 0.35
HPGD P15428 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP19A1 P11511 1/20 0.32
PGR P06401 2/20 0.32
AKR1C3 P42330 2/20 0.31
AKR1C2 P52895 2/20 0.31
SIGMAR1 Q99720 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
HCRTR1 O43613 1/20 0.30
SLC22A12 Q96S37 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5800554 0.98 PTGS2 (0.38) TSHRPTGS2HSD11B1HPGDALDH1A1
SCHEMBL5822674 0.94 PTGS2 (0.36) TSHRPTGS2CYP19A1AKR1C3AKR1C2
SCHEMBL5819680 0.92 PTGS2 (0.37) TSHRPTGS2CYP19A1AKR1C3AKR1C2
SCHEMBL5559333 0.90 PTGS2 (0.43) PTGS2AKR1C3AKR1C2
SCHEMBL5558388 0.90 PTGS2 (0.35) PTGS2HSD11B1ALDH1A1CYP19A1AKR1C3
SCHEMBL5819926 0.89 L3MBTL1 (0.37) TSHRPTGS2HSD11B1ALDH1A1
SCHEMBL5798701 0.89 PTGS2 (0.45) PTGS2CYP19A1AKR1C3AKR1C2
SCHEMBL5559153 0.88 TSHR (0.36) TSHRPTGS2HSD11B1HPGDALDH1A1
SCHEMBL5560260 0.88 PTGS2 (0.37) PTGS2HSD11B1HPGDALDH1A1CYP19A1
SCHEMBL5800993 0.87 PTGS2 (0.37) PTGS2HSD11B1ALDH1A1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed