SCHEMBL5819683

SCHEMBL5819683

CCc1ccc(-n2c(-c3ccc(SC)cc3)nc(=O)c(C(=N)NC)c2SC)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ATM Q13315 1/20 0.34
ALDH1A1 P00352 2/20 0.32
TP53 P04637 1/20 0.32
ESR1 P03372 1/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
TDP2 O95551 1/20 0.31
TNF P01375 1/20 0.30
HTT P42858 1/20 0.30
NOD2 Q9HC29 1/20 0.30
NOD1 Q9Y239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821767 0.93 ESR1 (0.36) SMN1; SMN2KDM4EALDH1A1ESR1PTGS1
SCHEMBL5820891 0.90 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1ESR1PTGS1PTGS2
SCHEMBL5815689 0.88 GRIA1 (0.36) ALDH1A1TP53ESR1PTGS1PTGS2
SCHEMBL5820973 0.86 ALDH1A1 (0.43) KDM4EALDH1A1HTT
SCHEMBL5820972 0.80 PTK2 (0.35) SMN1; SMN2KMT2AALDH1A1TP53PTGS2
SCHEMBL5821417 0.78 ALDH1A1 (0.36) MEN1KMT2AALDH1A1ESR1
SCHEMBL5819681 0.77 CA9 (0.43) KMT2AALDH1A1PTGS1PTGS2
SCHEMBL5822322 0.77 CA9 (0.43) KMT2AALDH1A1PTGS1PTGS2
SCHEMBL5821175 0.75 KMT2A (0.47) MEN1KMT2APTGS1PTGS2
SCHEMBL5815528 0.74 GAA (0.38) KMT2APTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO claimed