SCHEMBL5820972

SCHEMBL5820972

CNC(=N)c1c(SC)n(-c2cc(OC)c(OC)c(OC)c2)c(-c2ccc(SC)cc2)nc1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.35
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP1B1 Q16678 1/20 0.34
PTGS2 P35354 1/20 0.34
KATNA1 O75449 1/20 0.34
MAP3K11 Q16584 1/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
DHFR P00374 1/20 0.32
LMNA P02545 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPT P10636 3/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
PDGFRB P09619 1/20 0.31
KIT P10721 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821767 0.86 ESR1 (0.36) PTGS2SMN1; SMN2MAPTALDH1A1
SCHEMBL5820973 0.85 ALDH1A1 (0.43) NPC1RAB9ALMNAALDH1A1HTT
SCHEMBL5822048 0.85 PTK2 (0.35) PTK2CYP1A1CYP1A2CYP1B1PTGS2
SCHEMBL5820891 0.83 ALDH1A1 (0.41) PTGS2HPGDNPC1RAB9ADHFR
SCHEMBL5815689 0.81 GRIA1 (0.36) PTGS2ALDH1A1TP53RXFP1
SCHEMBL5819683 0.80 HCAR1 (0.34) PTGS2SMN1; SMN2ALDH1A1HTTKMT2A
SCHEMBL5821417 0.71 ALDH1A1 (0.36) LMNAMAPTALDH1A1KMT2A
SCHEMBL5819681 0.71 CA9 (0.43) PTGS2ALDH1A1KMT2A
SCHEMBL5822322 0.71 CA9 (0.43) PTGS2ALDH1A1KMT2A
SCHEMBL5821281 0.71 PTGS2 (0.38) PTGS2MAPTKMT2AKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed
WO-2006102674-A2 DIPHENYLHETEROCYCLE CHOLESTEROL ABSORPTION INHIBITORS MICROBIA, INC. (US) 2006-09-28 WO disclosed