SCHEMBL5820973

SCHEMBL5820973

CNC(=N)c1c(SC)n(-c2ccc(SC)cc2)c(-c2ccc(OC)cc2)nc1=O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
NPSR1 Q6W5P4 2/20 0.41
RAB9A P51151 2/20 0.41
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
GSK3B P49841 1/20 0.35
NPC1 O15118 2/20 0.34
MAPK1 P28482 1/20 0.34
GRM5 P41594 1/20 0.34
G6PD P11413 1/20 0.34
OXTR P30559 1/20 0.34
CNR1 P21554 3/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
CNR2 P34972 1/20 0.34
UBE2N P61088 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821767 0.93 ESR1 (0.36) ALDH1A1CNR1KDM4ECNR2
SCHEMBL5820891 0.90 ALDH1A1 (0.41) ALDH1A1NPSR1RAB9ALMNANPC1
SCHEMBL5815689 0.88 GRIA1 (0.36) ALDH1A1NPSR1GRM5
SCHEMBL5819683 0.86 HCAR1 (0.34) ALDH1A1KDM4EHTT
SCHEMBL5820972 0.85 PTK2 (0.35) ALDH1A1RAB9ALMNANPC1HTT
SCHEMBL5818323 0.85 G6PD (0.53) ALDH1A1LMNAMAPK1G6PDKDM4E
SCHEMBL5821417 0.78 ALDH1A1 (0.36) ALDH1A1LMNAGRM5
SCHEMBL5822322 0.77 CA9 (0.43) ALDH1A1
SCHEMBL5819681 0.77 CA9 (0.43) ALDH1A1
SCHEMBL5821175 0.75 KMT2A (0.47) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed