SCHEMBL5820740

SCHEMBL5820740

Cc1cc(CC(=O)NS(=O)(=O)c2ccc(Cl)s2)n(-c2ccccc2)n1.Cc1cc(CC(=O)NS(=O)(=O)c2ccc(F)cc2)n(-c2ccccc2)n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 1/20 0.43
HTT P42858 1/20 0.43
EGFR P00533 7/20 0.43
ERBB2 P04626 7/20 0.43
PTGES O14684 4/20 0.41
ALOX5 P09917 4/20 0.41
MAPT P10636 1/20 0.41
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5804793 0.90 AKR1C3 (0.40) ALDH1A1KDM4EHTTEGFRERBB2
SCHEMBL5820745 0.84 ALDH1A1 (0.44) ALDH1A1KDM4EHTTMAPTPOLB
SCHEMBL5809144 0.83 MAPT (0.46) ALDH1A1KDM4EHTTEGFRERBB2
SCHEMBL5807526 0.83 EGFR (0.58) ALDH1A1EGFRERBB2PTGESALOX5
SCHEMBL5807982 0.83 PTGES (0.56) ALDH1A1EGFRERBB2PTGESALOX5
SCHEMBL5804900 0.83 MAPK13 (0.47) ALDH1A1EGFRERBB2PTGESALOX5
SCHEMBL5806852 0.82 ALDH1A1 (0.50) ALDH1A1HTTEGFRERBB2PTGES
SCHEMBL5804485 0.81 EGFR (0.47) EGFRERBB2PTGESALOX5MAPK13
SCHEMBL5808774 0.81 ALDH1A1 (0.59) ALDH1A1EGFRERBB2PTGESALOX5
SCHEMBL5807701 0.81 MEN1 (0.41) ALDH1A1HTTMAPTPOLBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006075955-A1 PYRAZOLYL ACYLSULFONAMIDE DERIVATIVES AS ENDOTHELIN CONVERTING ENZYME INHIBITORS AND USEFUL IN THE TREATMENT OF CHRONIC OBSTRUCTIVE PULMONARY DISEASE ASTRAZENECA AB (SE) 2006-07-20 WO claimed