SCHEMBL5821054

SCHEMBL5821054

CNC(=N)c1c(NC)n(-c2ccc(OC)cc2)c(-c2cccnc2)nc1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
G6PD P11413 1/20 0.52
ALDH1A1 P00352 4/20 0.44
MAPT P10636 4/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPK1 P28482 2/20 0.41
HSD17B10 Q99714 1/20 0.41
HPGD P15428 2/20 0.41
CYP11B1 P15538 4/20 0.39
CYP11B2 P19099 4/20 0.39
TSHR P16473 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP17A1 P05093 1/20 0.39
KDM4E B2RXH2 1/20 0.38
THRB P10828 1/20 0.38
EGFR P00533 1/20 0.38
F12 P00748 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5818323 0.87 G6PD (0.53) G6PDALDH1A1MAPTMEN1KMT2A
SCHEMBL5816275 0.86 MAPT (0.44) G6PDMAPTMEN1KMT2AMAPK1
SCHEMBL5823518 0.85 G6PD (0.57) G6PDALDH1A1MAPTMEN1KMT2A
SCHEMBL5818138 0.81 G6PD (0.56) G6PDALDH1A1MAPTMEN1KMT2A
SCHEMBL5821115 0.80 ALDH1A1 (0.40) G6PDALDH1A1MAPTMEN1KMT2A
SCHEMBL5821439 0.72 CA9 (0.44) G6PDMAPTMEN1KMT2A
SCHEMBL5823523 0.72 G6PD (0.56) G6PDALDH1A1MAPTMEN1KMT2A
SCHEMBL5820973 0.71 ALDH1A1 (0.43) G6PDALDH1A1MAPK1CYP3A4KDM4E
SCHEMBL4637042 0.69 G6PD (0.57) G6PDALDH1A1MAPTMEN1KMT2A
SCHEMBL5821434 0.68 ALDH1A1 (0.42) G6PDALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed