SCHEMBL5821115

SCHEMBL5821115

CNNc1c(C(=N)NC)c(=O)nc(-c2ccncc2)n1-c1ccc(OC)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
G6PD P11413 1/20 0.38
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
MTOR P42345 1/20 0.36
PIK3CG P48736 1/20 0.36
TNKS2 Q9H2K2 6/20 0.35
PDE5A O76074 1/20 0.35
TNKS O95271 3/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
THRB P10828 1/20 0.35
NPC1 O15118 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821054 0.80 G6PD (0.52) ALDH1A1G6PDMAPTTHRBMAPK1
SCHEMBL5821434 0.77 ALDH1A1 (0.42) ALDH1A1RAB9ANPSR1G6PDPIK3CD
SCHEMBL5821030 0.74 GAA (0.31) ALDH1A1KMT2AGAA
SCHEMBL5820973 0.74 ALDH1A1 (0.43) ALDH1A1RAB9ANPSR1G6PDNPC1
SCHEMBL5818323 0.73 G6PD (0.53) ALDH1A1G6PDMAPTTHRBMAPK1
SCHEMBL5815685 0.71 AOC3 (0.41) ALDH1A1MAPTSMN1; SMN2CYP3A4CYP2C9
SCHEMBL5821417 0.71 ALDH1A1 (0.36) ALDH1A1MAPTMEN1KMT2A
SCHEMBL5823518 0.71 G6PD (0.57) ALDH1A1RAB9ANPSR1G6PDMAPT
SCHEMBL5818138 0.69 G6PD (0.56) ALDH1A1RAB9ANPSR1G6PDMAPT
SCHEMBL5815528 0.69 GAA (0.38) CYP2D6KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed