SCHEMBL5822256

SCHEMBL5822256

Nc1cc(Oc2ccc(-n3ccnc3)cc2)c(F)cc1[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICAM1 P05362 2/20 0.43
SELE P16581 2/20 0.43
VCAM1 P19320 2/20 0.43
MAPT P10636 3/20 0.41
LMNA P02545 2/20 0.41
SCN9A Q15858 1/20 0.40
PDE2A O00408 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
HTT P42858 1/20 0.38
NOS2 P35228 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP19A1 P11511 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1872393 0.77 CRHBP (0.45) VCAM1MAPTLMNAHSPB1
SCHEMBL8076008 0.76 GRIA1 (0.50) MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL16151007 0.76 MAPT (0.50) MAPTLMNAPDE2APDE3BPDE3A
SCHEMBL1067164 0.76 LMNA (0.52) MAPTLMNAPDE2APDE3BPDE3A
Hydrochloric Acid SCHEMBL8145134 0.75 GRIA1 (0.49) MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL5036730 0.74 CA1 (0.43) MAPTLMNAPDE2APDE3BPDE3A
SCHEMBL328169 0.73 HSPB1 (0.49) ICAM1SELEVCAM1MAPTLMNA
SCHEMBL2646431 0.73 SLC6A4 (0.43) VCAM1MAPTLMNASCN9ACYP1A2
SCHEMBL2644788 0.71 MAPT (0.45) VCAM1MAPTLMNAHTTCYP1A2
SCHEMBL15155950 0.70 HSPB1 (0.64) MAPTLMNAHTTCYP3A4HSPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663953-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-06-07 EP disclosed
WO-2005030705-A9 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC (CA) 2006-04-20 WO disclosed
WO-2005030704-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2005-04-07 WO disclosed
WO-2005030705-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2005-04-07 WO disclosed