SCHEMBL5822874

SCHEMBL5822874

NS(=O)(=O)c1ccc(-c2ccccc2-c2ncco2)cc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.54
PTGS1 P23219 3/20 0.54
CA2 P00918 14/20 0.50
CA1 P00915 12/20 0.50
CA9 Q16790 10/20 0.50
CA12 O43570 8/20 0.50
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
DRD1 P21728 1/20 0.47
IKBKB O14920 1/20 0.45
CHUK O15111 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547875 0.85 CA2 (0.45) PTGS2PTGS1CA2CA1CA9
SCHEMBL18118210 0.84 CA2 (0.54) CA2CA1CA9CA12MAOA
SCHEMBL9151503 0.80 LTA4H (0.46)
SCHEMBL6986037 0.79 EDNRB (0.56)
SCHEMBL9510279 0.79 HPGDS (0.58)
SCHEMBL7408116 0.79 BRD4 (0.41) CA2CA1CA9CA12
SCHEMBL6026444 0.78 BRD4 (0.43) CA2CA1CA9CA12
SCHEMBL7408121 0.78 HPGDS (0.44) PTGS2CA2CA1CA9CA12
SCHEMBL1919495 0.77 HPGDS (0.52)
SCHEMBL28477141 0.76 LTA4H (0.46) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006102898-A2 OXAPROZIN OR A CLOSELY RELATED COMPOUND FOR THE TREATMENT OF ECZEMA ASTION PHARMA A/S (DK) 2006-10-05 WO disclosed