SCHEMBL8547875

SCHEMBL8547875

NS(=O)(=O)c1ccc(-c2ccccc2)c(-c2ncco2)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.45
CA1 P00915 9/20 0.45
CA9 Q16790 8/20 0.45
CA13 Q8N1Q1 1/20 0.45
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
CA12 O43570 5/20 0.44
PTGS2 P35354 4/20 0.43
TDP1 Q9NUW8 1/20 0.43
HPGDS O60760 1/20 0.42
LRRK2 Q5S007 1/20 0.41
SCN9A Q15858 1/20 0.41
PTGS1 P23219 2/20 0.40
IKBKB O14920 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5822874 0.85 PTGS2 (0.54) CA2CA1CA9MAOAMAOB
SCHEMBL4733933 0.79 CA2 (0.61) CA2CA1CA9CA13CA12
SCHEMBL30069032 0.79 CA1 (0.57) CA2CA1CA9CA13MAOA
SCHEMBL18118203 0.79 CA1 (0.57) CA2CA1CA9CA13MAOA
SCHEMBL7129733 0.78 HPGDS (0.50) HPGDS
SCHEMBL8908994 0.78 MAOB (0.47) CA2CA1CA9MAOBCA12
SCHEMBL7408121 0.78 HPGDS (0.44) CA2CA1CA9CA13MAOA
SCHEMBL30434205 0.77 CA2 (0.64) CA2CA1CA9CA13CA12
SCHEMBL9510279 0.76 HPGDS (0.58) HPGDS
SCHEMBL942521 0.76 HPGDS (0.47) MAOBTDP1HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed