SCHEMBL5835618

SCHEMBL5835618

CCCC(=O)Nc1ncc(-c2ccccc2)s1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 1/20 0.69
CDK2 P24941 1/20 0.69
CDK5 Q00535 1/20 0.69
ACP1 P24666 1/20 0.66
KDR P35968 1/20 0.63
GSTO1 P78417 1/20 0.59
SCD O00767 1/20 0.58
ALDH1A1 P00352 2/20 0.57
MEN1 O00255 1/20 0.56
NPC1 O15118 1/20 0.56
LMNA P02545 1/20 0.56
RAB9A P51151 1/20 0.56
KMT2A Q03164 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
WNT3A P56704 1/20 0.56
CNR1 P21554 1/20 0.54
MKNK1 Q9BUB5 1/20 0.54
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962875 0.86 CCNE1 (0.66) CCNE1CDK2CDK5ACP1KDR
SCHEMBL69753 0.84 CCNE1 (0.74) CCNE1CDK2CDK5ACP1KDR
SCHEMBL70693 0.82 CCNE1 (0.63) CCNE1CDK2CDK5ACP1KDR
SCHEMBL5840422 0.81 KDR (0.72) CCNE1CDK2CDK5ACP1KDR
SCHEMBL21484795 0.80 CCNE1 (0.67) CCNE1CDK2CDK5ACP1KDR
SCHEMBL5835965 0.78 LMNA (0.65) CCNE1CDK2CDK5ALDH1A1MEN1
SCHEMBL21962874 0.78 KDR (0.60) CCNE1CDK2CDK5ACP1KDR
SCHEMBL17014785 0.78 KDR (0.68) CCNE1CDK2CDK5ACP1KDR
SCHEMBL10252594 0.78 KDR (1.00) CCNE1CDK2CDK5ACP1KDR
SCHEMBL2256136 0.78 KDR (0.72) CCNE1CDK2CDK5ACP1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1325389-A 2-aminothiazole derivatives, process for preparing the same and their use as antitumor agents PHARMACIA & UPJOHN SPA (IT) 2001-12-05 CN claimed
US-7037929-B1 2-amino-thiazole derivatives, process for their preparation, and their use as antitumor agents PHARMACIA & UPJOHN S.P.A. (IT) 2006-05-02 US disclosed
CN-1325389-A 2-aminothiazole derivatives, process for preparing the same and their use as antitumor agents PHARMACIA & UPJOHN SPA (IT) 2001-12-05 CN disclosed