SCHEMBL5840339

SCHEMBL5840339

CCOC(=O)c1cccc(Nc2nc(Cl)nc3nc[nH]c23)c1C

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.52
TNNI3K Q59H18 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 1/20 0.45
XDH P47989 1/20 0.44
CDC25A P30304 1/20 0.44
CDC25B P30305 1/20 0.44
CDC25C P30307 1/20 0.44
TMIGD3 P0DMS9 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5840336 0.85 MAPT (0.43) SMN1; SMN2KDM4ETP53KMT2ACDC25A
SCHEMBL5839549 0.75 YTHDC1 (0.46) NPC1CDC25ACDC25BCDC25C
SCHEMBL28724597 0.73 KDM4E (0.47) BRAFSMN1; SMN2KDM4ENPC1TP53
SCHEMBL29696548 0.73 KDM4E (0.47) BRAFSMN1; SMN2KDM4ENPC1TP53
SCHEMBL3007044 0.72 BRAF (0.72) BRAFTNNI3KSMN1; SMN2XDHTMIGD3
SCHEMBL7788943 0.72 TNNI3K (0.62) BRAFTNNI3K
SCHEMBL31344585 0.70 XDH (0.52) BRAFTNNI3KSMN1; SMN2XDHTMIGD3
SCHEMBL1203877 0.70 METTL3 (0.56) SMN1; SMN2KDM4ETP53HPGDCDC25A
SCHEMBL1203237 0.70 METTL3 (0.56) SMN1; SMN2KDM4ETP53HPGDKMT2A
SCHEMBL17916012 0.70 AURKA (0.47) SMN1; SMN2NPC1TP53RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091346-B1 Purine derivatives and processes for their preparation NOVARTIS AG (CH) 2006-08-15 US disclosed
EP-0874846-B1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 2003-04-02 EP disclosed
CN-1066147-C Purine derivatives and process for preparing same 诺瓦提斯公司 2001-05-23 CN disclosed
CN-1202896-A Purine derivatives and processes for their preparation 诺瓦提斯公司 1998-12-23 CN disclosed
EP-0874846-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION Novartis AG (CH) 1998-11-04 EP disclosed
WO-1997016452-A1 PURINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1997-05-09 WO disclosed