SCHEMBL5847306

SCHEMBL5847306

CCOc1ccc(-c2cc3c4c(c2C(C)(C)C)[C@@H]2CN(C(=O)O)CC[C@@H]2N4CC3)c(C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
RBP4 P02753 1/20 0.32
MCHR1 Q99705 1/20 0.32
EPHX2 P34913 3/20 0.31
MAPT P10636 2/20 0.31
ACHE P22303 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
NPY2R P49146 1/20 0.31
LIPE Q05469 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
KMT2A Q03164 1/20 0.30
HSD11B1 P28845 1/20 0.30
CPT2 P23786 1/20 0.30
CPT1A P50416 1/20 0.30
FFAR1 O14842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847800 0.91 HTR2A (0.44) HTR2AHTR2CHTR2BRBP4EPHX2
SCHEMBL5847475 0.90 S1PR1 (0.37) HTR2AHTR2CHTR2BEPHX2
SCHEMBL5847107 0.85 SCD5 (0.37) HTR2AHTR2CHTR2BRBP4MCHR1
SCHEMBL5410829 0.84 HTR2A (0.51) HTR2AHTR2CHTR2BRBP4MCHR1
SCHEMBL5847619 0.81 CPS1 (0.37) HTR2AHTR2CHTR2B
SCHEMBL5847121 0.80 CCR3 (0.35) HTR2AHTR2CHTR2BMCHR1ALDH1A1
SCHEMBL5846973 0.80 CCR3 (0.34) HTR2AHTR2CHTR2BMCHR1
SCHEMBL5847193 0.79 CCR3 (0.35) HTR2AHTR2CHTR2BKMT2A
SCHEMBL5847324 0.79 CCR3 (0.34) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL5847854 0.78 HCRTR1 (0.36) HTR2AHTR2CEPHX2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed