SCHEMBL5847222

SCHEMBL5847222

CCC(=O)OC([O])C(O)CO

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP2C19 P33261 1/20 0.34
RECQL P46063 1/20 0.34
USP2 O75604 1/20 0.33
SLCO1B1 Q9Y6L6 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
PDE4A P27815 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 2/20 0.31
KDM4E B2RXH2 1/20 0.31
DUSP3 P51452 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847228 0.83 ALDH1A1 (0.43) MEN1KMT2AUSP2MAPTMAPK1
SCHEMBL9698326 0.81 MEN1 (0.33) MEN1KMT2ACYP2C19RECQLMAPT
SCHEMBL18877228 0.80 MEN1 (0.35) MEN1KMT2ACYP2C19RECQLUSP2
SCHEMBL4616283 0.77 MEN1 (0.33) MEN1KMT2ACYP2C19RECQLMAPT
SCHEMBL10500851 0.77 MEN1 (0.33) MEN1KMT2ACYP2C19RECQLMAPT
SCHEMBL12475543 0.77 MEN1 (0.33) MEN1KMT2ACYP2C19RECQLMAPT
SCHEMBL9638912 0.77 MAPT (0.36) MEN1KMT2ACYP2C19RECQLMAPT
SCHEMBL4624024 0.76 MEN1 (0.31) MEN1KMT2ACYP2C19RECQLMAPT
SCHEMBL18877226 0.75 LMNA (0.39) MEN1KMT2ACYP2C19RECQLUSP2
SCHEMBL7528074 0.75 MEN1 (0.33) MEN1KMT2ACYP2C19RECQLMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040023805-A1 Substituted phenyluracils ANDREE ROLAND (DE) 2004-02-05 US claimed
US-6649760-B2 Herbicides BAYER AKTIENGESELLSCHAFT (DE) 2003-11-18 US claimed
US-20020173425-A1 Substituted phenyluracils BAYER AKTIENGESELLSCHAFT (DE) 2002-11-21 US claimed
EP-0759908-A1 SUBSTITUTED DIAZACYCLOHEXANDI(THI)ONES BAYER AG (DE) 1997-03-05 EP claimed
WO-1995031440-A1 SUBSTITUTED DIAZACYCLOHEXANDI(THI)ONES BAYER AKTIENGESELLSCHAFT (DE) 1995-11-23 WO claimed
EP-0251294-B1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND ANTI-ULCER AGENTS SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1990-09-19 EP claimed
EP-0112191-B1 4-(1H-INDOLYL-3-)-ALPHA-METHYL PIPERIDINE-1-ETHANOL DERIVATIVES, THEIR SALTS, PROCESS FOR THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND THEIR USE AS MEDICINES ROUSSEL-UCLAF (FR) 1987-02-04 EP claimed
US-6992044-B1 Substituted phenyluracils BAYER CROPSCIENCE AG (DE) 2006-01-31 US disclosed
US-20040023805-A1 Substituted phenyluracils ANDREE ROLAND (DE) 2004-02-05 US disclosed
US-6649760-B2 Herbicides BAYER AKTIENGESELLSCHAFT (DE) 2003-11-18 US disclosed
US-20020173425-A1 Substituted phenyluracils BAYER AKTIENGESELLSCHAFT (DE) 2002-11-21 US disclosed
US-6429203-B1 PHOSPHOSESQUITERPENES USED TO TREAT CANCER; REDUCED SIDE EFFECTS INTERNATIONAL PHYTOCHEMISTRY RESEARCH LABS, LTD. 2002-08-06 US disclosed
US-6268394-B1 CONTACTING A CELL WITH AN AMOUNT OF A SESQUITERPENE LACTONE INTERNATIONAL PHYTOCHEMISTRY RESEARCH LABS, LTD. 2001-07-31 US disclosed
EP-1056450-A1 FARNESYL-PROTEIN TRANSFERASE INHIBITORS International Phytochemistry Research Labs, Ltd. (US) 2000-12-06 EP disclosed
US-6150375-A INHIBITORS OF BOTH OF THE HUMAN 5AR ISOZYMES; BENIGN PROSTATE HYPERPLASIA, MALE PATTERN BALDNESS, ACNE VULGARIS, SEBORRHEA, ANDROGENIC ALOPECIA, HIRSUTISM AND PROSTATE CANCER; BLOCKS THE CONVERSION OF TESTOSTERONE TO 5-ALPHA-DIHYDROTESTOSTERONE ELI LILLY AND COMPANY (US) 2000-11-21 US disclosed
US-6051565-A Farnesyl-protein transferase inhibitors INTERNATIONAL PHYTOCHEMISTRY RESEARCH LABS, LTD. (US) 2000-04-18 US disclosed
WO-1999043314-A1 FARNESYL-PROTEIN TRANSFERASE INHIBITORS INTERNATIONAL PHYTOCHEMISTRY RESEARCH LABS, LTD. (US) 1999-09-02 WO disclosed
EP-0358118-B1 Phenylamides - process for their preparation as well as a drug containing those compounds BOEHRINGER MANNHEIM GMBH (DE) 1994-03-16 EP disclosed
EP-0358118-A1 Phenylamides - process for their preparation as well as a drug containing those compounds Roche Diagnostics GmbH (DE) 1990-03-14 EP disclosed
EP-0251998-A2 Phenylsulfonylureas CIBA-GEIGY AG (CH) 1988-01-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020173425-A1 Substituted phenyluracils DPYD, POP1, G6PD MEN1 3334/4885KMT2A 1862/4885CYP2C19 429/4885
US-20040023805-A1 Substituted phenyluracils DPYD, POP1, G6PD MEN1 3334/4885KMT2A 1862/4885CYP2C19 429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.