SCHEMBL5848064

SCHEMBL5848064

CC(C)(C)c1c(-c2ccc(Cl)cc2F)cc2c3c1[C@@H]1CN(C(=O)O)CC[C@@H]1N3CC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
PDK2 Q15119 2/20 0.33
USP30 Q70CQ3 1/20 0.33
GRM2 Q14416 2/20 0.31
OPRL1 P41146 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CCR3 P51677 1/20 0.31
MAP4K4 O95819 1/20 0.31
EGFR P00533 1/20 0.31
PRKACA P17612 1/20 0.31
FRK P42685 1/20 0.31
MAPK9 P45984 1/20 0.31
CSNK1A1 P48729 1/20 0.31
CSNK1D P48730 1/20 0.31
MINK1 Q8N4C8 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
MC4R P32245 3/20 0.30
MC5R P33032 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848598 0.89 TSHR (0.33) DPP4DPP7CCR3
SCHEMBL5847619 0.88 CPS1 (0.37) CCR3
SCHEMBL5848396 0.85 CCR3 (0.31) CCR3
SCHEMBL5847854 0.83 HCRTR1 (0.36) DPP4DPP7CCR3
SCHEMBL5847193 0.82 CCR3 (0.35) PDK2CCR3FASN
SCHEMBL5849715 0.82 DRD1 (0.37) DPP4DPP7CCR3
SCHEMBL5847392 0.82 CCR3 (0.34) CCR3
SCHEMBL5847107 0.81 SCD5 (0.37) DPP4DPP7CCR3
SCHEMBL5849356 0.80 CCR3 (0.30) CCR3
SCHEMBL5413163 0.80 CCR3 (0.36) DPP4DPP7CCR3FASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed