SCHEMBL5860145

SCHEMBL5860145

COC1=C(OC)C(=O)C(c2cc(C)c(-c3cccnc3)c(C(=O)Nc3ccc(OC)cc3)c2)=C(C)C1=O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.49
PSMD14 O00487 1/20 0.49
IRAK4 Q9NWZ3 1/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 1/20 0.47
ATR Q13535 1/20 0.46
ABL1 P00519 3/20 0.45
BCR P11274 1/20 0.45
LMNA P02545 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PKM P14618 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
KDR P35968 1/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5859281 0.90 CYP3A4 (0.48) BRAFKMT2APOLBLMNAPKM
SCHEMBL5859923 0.90 MAPT (0.49) BRAFKMT2AABL1BCRLMNA
SCHEMBL5859855 0.89 NPC1 (0.51) KMT2APOLBLMNARAB9ANPC1
SCHEMBL5862046 0.89 NPC1 (0.50) KMT2APOLBLMNAKDM4ERAB9A
SCHEMBL5859069 0.87 NPC1 (0.46) KMT2APOLBLMNAKDM4ERAB9A
SCHEMBL5859192 0.85 PSMD14 (0.51) BRAFPSMD14IRAK4KMT2APOLB
SCHEMBL5862147 0.83 KDM4E (0.42) LMNAKDM4E
SCHEMBL5859082 0.81 MEN1 (0.48) KMT2APOLBLMNARAB9ANPC1
SCHEMBL5860337 0.80 APOB (0.44) BRAF
SCHEMBL5859235 0.77 CYP2C9 (0.45) KMT2AABL1BCRTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122543-B2 Substituted benzoic acid derivatives having NF-κB inhibiting action DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2006-10-17 US disclosed
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed