SCHEMBL5860337

SCHEMBL5860337

COC1=C(OC)C(=O)C(c2cc(C)c(-c3ccncc3)c(C(=O)Nc3ccc(C(F)(F)F)cc3)c2)=C(C)C1=O

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
APOB P04114 10/20 0.44
MTTP P55157 10/20 0.44
SMO Q99835 4/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
TRPV1 Q8NER1 3/20 0.42
BRAF P15056 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5859923 0.91 MAPT (0.49) TRPV1BRAF
SCHEMBL5859281 0.90 CYP3A4 (0.48) JAK2TYK2BRAF
SCHEMBL5860306 0.86 SMO (0.44) APOBMTTPSMOJAK2JAK1
SCHEMBL5862046 0.83 NPC1 (0.50)
SCHEMBL5859855 0.81 NPC1 (0.51)
SCHEMBL5859860 0.80 IKBKB (0.37)
SCHEMBL5860145 0.80 BRAF (0.49) BRAF
SCHEMBL5859140 0.79 CNR1 (0.45) TYK2
SCHEMBL5859286 0.79 TAS1R3 (0.38)
SCHEMBL6661408 0.78 GPR27 (0.44) APOBMTTPSMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122543-B2 Substituted benzoic acid derivatives having NF-κB inhibiting action DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2006-10-17 US disclosed
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed