SCHEMBL5862046

SCHEMBL5862046

COC1=C(OC)C(=O)C(c2cc(C)c(-c3ccc(OC)cc3)c(C(=O)Nc3ccc(OC)cc3)c2)=C(C)C1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.50
RAB9A P51151 2/20 0.50
LMNA P02545 2/20 0.47
KDR P35968 1/20 0.47
ALDH1A1 P00352 3/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
CASP3 P42574 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
METAP2 P50579 1/20 0.43
MAOB P27338 1/20 0.43
PSMB11 A5LHX3 1/20 0.42
PSMA7 O14818 1/20 0.42
PSMB1 P20618 1/20 0.42
PSMA1 P25786 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5859855 0.96 NPC1 (0.51) NPC1RAB9ALMNAKDRALDH1A1
SCHEMBL5859281 0.93 CYP3A4 (0.48) NPC1RAB9ALMNAKDRALDH1A1
SCHEMBL5859069 0.92 NPC1 (0.46) NPC1RAB9ALMNAKDRALDH1A1
SCHEMBL5860145 0.89 BRAF (0.49) NPC1RAB9ALMNAKDRMAPT
SCHEMBL5859082 0.88 MEN1 (0.48) NPC1RAB9ALMNAKDRALDH1A1
SCHEMBL5862164 0.85 GPR35 (0.44) NPC1RAB9ALMNAALDH1A1MAPT
SCHEMBL5860337 0.83 APOB (0.44)
SCHEMBL5859859 0.78 TDP1 (0.46) NPC1RAB9ALMNAALDH1A1HPGD
SCHEMBL7064963 0.78 POLB (0.44) NPC1RAB9AALDH1A1MAPTMEN1
SCHEMBL5859923 0.78 MAPT (0.49) LMNAKDRMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122543-B2 Substituted benzoic acid derivatives having NF-κB inhibiting action DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2006-10-17 US disclosed
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed