SCHEMBL5864155

SCHEMBL5864155

CCOC(=O)c1cccc(N2CCN(CCC(c3ccc(Cl)cc3)c3ccc(Cl)cc3)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.51
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
MAPK1 P28482 1/20 0.48
KMT2A Q03164 1/20 0.48
HTR1A P08908 4/20 0.46
KCNA3 P22001 1/20 0.46
HTR7 P34969 1/20 0.45
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
ENPP2 Q13822 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5863895 0.92 KCNA3 (0.54) MAPTLMNAKCNA3HTR7ALDH1A1
SCHEMBL5864102 0.90 SLC6A2 (0.48) MAPTMEN1LMNAKMT2AHTR1A
SCHEMBL6420684 0.81 ALOX5 (0.52) MAPTMEN1LMNAMAPK1KMT2A
SCHEMBL6707329 0.79 PRMT1 (0.67) MAPTMEN1LMNAMAPK1KMT2A
SCHEMBL8698788 0.78 PLOD2 (0.56) MAPTMEN1LMNAMAPK1KMT2A
Iodide SCHEMBL6706501 0.78 PRMT1 (0.66) MAPTMEN1LMNAMAPK1KMT2A
SCHEMBL5863335 0.77 KDM4E (0.57) MEN1KMT2AKCNA3HTR7DRD2
SCHEMBL5863375 0.77 HTR2C (0.46) LMNAHTR1ADRD4ALDH1A1
SCHEMBL3189295 0.77 HTR7 (0.50) MAPTLMNAMAPK1HTR1AHTR7
SCHEMBL3189302 0.77 KCNH2 (0.51) MAPTLMNAHTR7DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030120-B2 Nitrogen-containing heterocyclic compounds and benzamide compounds and drugs containing the same MEIJI SEIKA KAISHA, LTD. (JP) 2006-04-18 US disclosed
US-20040224959-A1 Nitrogen-containing heterocyclic compounds and benzamide compounds and drugs containing the same OHKURA NAOTO (JP) 2004-11-11 US disclosed
US-6777414-B1 INHIBITORS OF TRIGLYCERIDE BIOSYNTHESIS AND SECRETION OF APOLIPOPROTEIN B-CONTAINING LIPOPROTEINS; ARTERIOSCLEROTIC DISEASES; HYPERLIPIDEMIA MEIJI SEIKA KAISHA, LTD. (JP) 2004-08-17 US disclosed
EP-1180514-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND BENAMIDE COMPOUNDS AND DRUGS CONTAINING THE SAME MEIJI SEIKA KAISHA LTD. (JP) 2002-02-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040224959-A1 Nitrogen-containing heterocyclic compounds and benzamide compounds and drugs containing the same APOB, NCEH1, LIPC MAPT 4733/4885MEN1 4072/4885LMNA 508/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.