SCHEMBL5867018

SCHEMBL5867018

CS(=O)(=O)Nc1cccc2cc(C(=Nc3cccc(Cl)c3)NO)oc12

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 10/20 0.42
LMNA P02545 1/20 0.40
CRHR1 P34998 5/20 0.38
NR3C1 P04150 2/20 0.38
KEAP1 Q14145 1/20 0.38
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
AR P10275 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
GLO1 Q04760 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5867013 0.79 CTPS1 (0.42) LMNANR3C1KEAP1HTT
SCHEMBL5867011 0.79 CTPS1 (0.42) LMNANR3C1KEAP1HTT
SCHEMBL5867090 0.79 IDO1 (0.52) IDO1LMNA
SCHEMBL5935553 0.78 LMNA (0.53) IDO1LMNAHTT
SCHEMBL5866943 0.74 KCNQ2 (0.43) IDO1LMNAHTT
SCHEMBL6777820 0.73 KEAP1 (0.40) LMNANR3C1KEAP1PGRNR3C2
SCHEMBL5866921 0.73 IDO1 (0.62) IDO1LMNA
SCHEMBL5866888 0.70 LMNA (0.52) IDO1LMNACRHR1
SCHEMBL5866857 0.69 IDO1 (0.58) IDO1
SCHEMBL5866850 0.67 LMNA (0.62) IDO1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7148259-B1 Antibacterial agents AMGEN INC. (US) 2006-12-12 US disclosed
US-20060270651-A1 ANTIBACTERIAL AGENTS AMGEN INC. (US) 2006-11-30 US disclosed
US-7053234-B2 Antibacterial agents AMGEN INC. (US) 2006-05-30 US disclosed
US-20040235911-A1 hydroxyamidines; antibiotic resistance TULARIK INC. 2004-11-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040235911-A1 hydroxyamidines; antibiotic resistance HNMT, HDHD5, ABCC1 IDO1 3464/4885LMNA 4115/4885CRHR1 4539/4885
US-20060270651-A1 ANTIBACTERIAL AGENTS MRPL21, HDHD5, CLPP IDO1 3821/4885LMNA 4203/4885CRHR1 4799/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.