SCHEMBL5867429

SCHEMBL5867429

O=Cc1ccc(Br)cc1.OB(O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.59
KDM4E B2RXH2 1/20 0.59
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
TSHR P16473 1/20 0.50
TRPV6 Q9H1D0 2/20 0.46
ORAI1 Q96D31 1/20 0.46
ORAI2 Q96SN7 1/20 0.46
ORAI3 Q9BRQ5 1/20 0.46
HDAC3 O15379 1/20 0.41
ADAM17 P78536 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
GPR183 P32249 1/20 0.40
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5867390 0.81 KDM4E (0.51) MGLLKDM4ECA1CA2TRPV6
SCHEMBL5867371 0.80 MGLL (0.53) MGLLKDM4ECA1CA2TSHR
Tolyl Boronic Acid SCHEMBL27517807 0.79 KDM4E (0.66) KDM4ECA1CA2TSHRTRPV6
Trifluoromethylbenzene SCHEMBL28839038 0.78 ALDH1A1 (0.52) TSHRHDAC3ADAM17HDAC1HDAC2
SCHEMBL4179 0.77 MGLL (1.00) MGLLCA1CA2TSHRTRPV6
SCHEMBL61631 0.77 CYP1A2 (0.54) CA1CA2TSHRHDAC3ADAM17
SCHEMBL5840 0.77 KDM4E (1.00) KDM4ECA1CA2TSHR
Formic Acid SCHEMBL31514292 0.75 CES2 (0.46) MGLLCA1CA2TRPV6ORAI1
Methane SCHEMBL28841002 0.75 KDM4E (0.95) KDM4ECA1CA2TSHR
Hydrochloric Acid SCHEMBL27615734 0.75 CYP1A2 (0.52) CA1CA2HDAC3ADAM17HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115616-B2 Pyrimidinone compounds SMITHKLINE BEECHAM PLC (GB) 2006-10-03 US disclosed