SCHEMBL586902

SCHEMBL586902

CCOC(=O)CC(=O)[C@@H]1CCN(C)[C@H](C(F)c2cc(F)cc(F)c2)C1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.38
ALDH1A1 P00352 4/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CCL5 P13501 1/20 0.33
CCR5 P51681 1/20 0.33
CHRM3 P20309 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL587020 0.87 CHRM1 (0.37) CHRM1ALDH1A1TDP1MAPTKDM4E
SCHEMBL582160 0.74 KMT2A (0.41) CHRM1ALDH1A1TDP1KDM4EKMT2A
SCHEMBL582882 0.73 ALDH1A1 (0.44) ALDH1A1TDP1KDM4EKMT2ACHRM3
SCHEMBL582364 0.73 HTR2A (0.41) CHRM1ALDH1A1KMT2AL3MBTL1
SCHEMBL3085316 0.72 CHRM1 (0.38) CHRM1ALDH1A1TDP1MAPTKDM4E
SCHEMBL581176 0.72 CHRM1 (0.38) CHRM1ALDH1A1TDP1MAPTKDM4E
SCHEMBL3069035 0.72 CHRM1 (0.38) CHRM1ALDH1A1TDP1MAPTKDM4E
SCHEMBL586931 0.72 KDM4E (0.39) ALDH1A1TDP1MAPTKDM4EKMT2A
SCHEMBL580903 0.70 GAA (0.36) CHRM1ALDH1A1MAPTKDM4EL3MBTL1
SCHEMBL581244 0.70 GAA (0.36) CHRM1ALDH1A1MAPTKDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed