SCHEMBL5870467

SCHEMBL5870467

COC(=O)[C@H]1COC(=O)N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
CYP2D6 P10635 2/20 0.35
EGFR P00533 2/20 0.33
BRD4 O60885 1/20 0.33
BACE1 P56817 1/20 0.33
CHRNB2 P17787 2/20 0.32
CHRNA4 P43681 2/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA7 P36544 1/20 0.32
CYP1A2 P05177 2/20 0.32
HIF1A Q16665 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3135126 1.00 KMT2A (0.44) KMT2ACYP2D6EGFRBRD4BACE1
SCHEMBL3135120 1.00 KMT2A (0.44) KMT2ACYP2D6EGFRBRD4BACE1
SCHEMBL31590369 1.00 KMT2A (0.44) KMT2ACYP2D6EGFRBRD4BACE1
SCHEMBL21584101 0.81 KMT2A (0.41) KMT2ACYP2D6BRD4BACE1CHRNB2
SCHEMBL13439593 0.81 KMT2A (0.41) KMT2ACYP2D6BRD4BACE1CHRNB2
SCHEMBL31073506 0.80 ALDH1A1 (0.37) KMT2ACYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL3633924 0.80 ALDH1A1 (0.37) KMT2ACYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL5877457 0.79 KMT2A (0.39) KMT2ABACE1CHRNB2CHRNA4CHRNB4
SCHEMBL5877461 0.79 KMT2A (0.39) KMT2ABACE1CHRNB2CHRNA4CHRNB4
SCHEMBL6186602 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250114369-A1 COMPOUNDS AND METHODS FOR TREATMENT OF VIRAL INFECTIONS GILEAD SCIENCES, INC. 2025-04-10 US disclosed
WO-2025059427-A1 COMPOUNDS AND METHODS FOR TREATMENT OF VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2025-03-20 WO disclosed
CN-114031572-A Process for preparing substituted cycloserines 先正达参股股份有限公司 2022-02-11 CN disclosed
US-20180319800-A1 (1R,4R) 7-OXO-2-AZABICYCLO[2.2.2]OCT-5-ENE AND DERIVATIVES THEREOF DEMERX, INC. (US) 2018-11-08 US disclosed
US-10112931-B2 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH NOVARTIS AG (CH) 2018-10-30 US disclosed
US-20180051015-A1 3-PYRIMIDIN-4-YL-OXAZOLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH NOVARTIS AG (CH) 2018-02-22 US disclosed
EP-2970240-B1 3-PYRIMIDIN-4-YL-OXAZOLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH NOVARTIS AG (CH) 2018-01-10 EP disclosed
US-9839641-B2 Compounds and methods for treating bacterial infections ENTASIS THERAPEUTICS LIMITED (GB) 2017-12-12 US disclosed
US-9839641-B2 Compounds and methods for treating bacterial infections ENTASIS THERAPEUTICS LIMITED (GB) 2017-12-12 US disclosed
US-9688672-B2 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH NOVARTIS AG (CH) 2017-06-27 US disclosed
US-8889671-B2 Compounds and methods for treating bacterial infections ASTRAZENECA AB (SE) 2014-11-18 US disclosed
US-8889671-B2 Compounds and methods for treating bacterial infections ASTRAZENECA AB (SE) 2014-11-18 US disclosed
US-20140275083-A1 3-PYRIMIDIN-4-YL-OXAZOLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH NOVARTIS AG (CH) 2014-09-18 US disclosed
WO-2014141104-A1 3-PYRIMIDIN-4-YL-OXAZOLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH NOVARTIS AG (CH) 2014-09-18 WO disclosed
US-20140206677-A1 COMPOUNDS AND METHODS FOR TREATING BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2014-07-24 US disclosed
US-20140206677-A1 COMPOUNDS AND METHODS FOR TREATING BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2014-07-24 US disclosed
US-20130267710-A1 (1R,4R) 7-OXO-2-AZABICYCLO[2.2.2]OCT-5-ENE AND DERIVATIVES THEREOF DEMERX, INC. 2013-10-10 US disclosed
US-7045532-B2 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-05-16 US disclosed
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. 2004-04-29 US disclosed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140206677-A1 COMPOUNDS AND METHODS FOR TREATING BACTERIAL INFECTIONS NISCH, ELANE, ALPI KMT2A 4669/4885CYP2D6 271/4885EGFR 1668/4885
US-20130267710-A1 (1R,4R) 7-OXO-2-AZABICYCLO[2.2.2]OCT-5-ENE AND DERIVATIVES THEREOF AZI2, CYP4B1, OXER1 KMT2A 1282/4885CYP2D6 99/4885EGFR 2583/4885
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof ACE, ACE2, AGTR2 KMT2A 1880/4885CYP2D6 607/4885EGFR 3370/4885
US-20140275083-A1 3-PYRIMIDIN-4-YL-OXAZOLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH IDH1, IDH3B, IDH3A KMT2A 78/4885CYP2D6 1682/4885EGFR 477/4885
US-20180051015-A1 3-PYRIMIDIN-4-YL-OXAZOLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH IDH1, IDH3B, IDH3A KMT2A 78/4885CYP2D6 1682/4885EGFR 477/4885
US-20180319800-A1 (1R,4R) 7-OXO-2-AZABICYCLO[2.2.2]OCT-5-ENE AND DERIVATIVES THEREOF AZI2, CYP4B1, OXER1 KMT2A 1282/4885CYP2D6 99/4885EGFR 2583/4885
US-20250114369-A1 COMPOUNDS AND METHODS FOR TREATMENT OF VIRAL INFECTIONS HAVCR2, EIF2AK2, RPL35 KMT2A 3809/4885CYP2D6 817/4885EGFR 2208/4885
US-10112931-B2 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH IDH1, IDH3B, IDH3A KMT2A 78/4885CYP2D6 1682/4885EGFR 477/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.