SCHEMBL587150

SCHEMBL587150

COC(=O)C1CCN(C(=O)OC)C(CC2CCC(F)(F)CC2)C1.COC(=O)N1CCC(C(=O)O)CC1CC1CCC(F)(F)CC1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.33
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
IL1B P01584 3/20 0.33
P2RX7 Q99572 2/20 0.33
ALDH1A1 P00352 3/20 0.32
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
EPHX2 P34913 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL580791 0.95 BRD4 (0.34) BRD4CREBBPIL1BP2RX7EPHX2
SCHEMBL3073995 0.95 OPRK1 (0.35) OPRK1IL1BP2RX7ALDH1A1MAPT
SCHEMBL586873 0.82 IL1B (0.30) IL1BP2RX7
SCHEMBL581808 0.81 ALDH1A1 (0.39) BRD4CREBBPALDH1A1MAPTHSD17B10
SCHEMBL581649 0.80 GAA (0.32) IL1BP2RX7ALDH1A1MAPTGAA
SCHEMBL582194 0.80 GAA (0.32) IL1BP2RX7ALDH1A1MAPTGAA
SCHEMBL3078365 0.80 GAA (0.32) IL1BP2RX7ALDH1A1MAPTGAA
SCHEMBL1287034 0.75 OPRK1 (0.34) OPRK1
SCHEMBL1287102 0.75 OPRK1 (0.42) OPRK1ALDH1A1MAPTNPSR1HPGD
SCHEMBL580419 0.73 RAB9A (0.37) ALDH1A1MAPTNPSR1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed