SCHEMBL587575

SCHEMBL587575

COC(=O)C1CCN(C(=O)OC)C(c2ccc(S(C)(=O)=O)cc2)C1.COC(=O)N1CCC(C(=O)O)CC1c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.43
PKM P14618 1/20 0.41
MMP1 P03956 2/20 0.40
ADAM17 P78536 2/20 0.40
TP53 P04637 1/20 0.39
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
EPHX2 P34913 1/20 0.36
APEX1 P27695 1/20 0.36
PTGS2 P35354 2/20 0.36
HCRTR2 O43614 1/20 0.36
RIPK1 Q13546 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NR1H2 P55055 3/20 0.35
NR1H3 Q13133 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL580914 0.96 SLC6A4 (0.42) SLC6A4PKMALDH1A1EPHX2APEX1
SCHEMBL586843 0.96 SLC6A4 (0.47) SLC6A4PKMMMP1ADAM17TP53
SCHEMBL587433 0.85 SMN1; SMN2 (0.44) SLC6A4MAPT
SCHEMBL587349 0.85 MMP1 (0.41) SLC6A4MMP1ADAM17
SCHEMBL582439 0.84 ALDH1A1 (0.36) SLC6A4PKMALDH1A1NPSR1HPGD
SCHEMBL582438 0.84 ALDH1A1 (0.36) SLC6A4PKMALDH1A1NPSR1HPGD
SCHEMBL580837 0.84 RIPK1 (0.41) SLC6A4ALDH1A1EPHX2APEX1PTGS2
SCHEMBL586674 0.83 NOTUM (0.44) ALDH1A1MAPT
SCHEMBL582040 0.82 ALDH1A1 (0.48) SLC6A4ALDH1A1MAPTNPSR1HPGD
SCHEMBL586614 0.82 ALDH1A1 (0.43) SLC6A4PKMMMP1ADAM17TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed