SCHEMBL5877102

SCHEMBL5877102

Cc1ccc2nc(-c3ccc(-c4cccs4)s3)n(CC3CCCC(CN)C3)c(=O)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ADORA1 P30542 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
PLA2G1B P04054 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
ABCC1 P33527 1/20 0.37
AVPR1B P47901 1/20 0.36
GHSR Q92847 3/20 0.36
CYP2D6 P10635 2/20 0.36
HTR2C P28335 1/20 0.36
CYP3A4 P08684 1/20 0.35
KCNH2 Q12809 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486076 0.91 CYP2D6 (0.40) ALDH1A1KDM4EADORA1SMN1; SMN2MEN1
SCHEMBL5877351 0.90 AVPR1B (0.40) ALDH1A1ADORA1MEN1LMNAHPGD
SCHEMBL5877833 0.89 ABCC1 (0.45) ALDH1A1KDM4EADORA1SMN1; SMN2MEN1
SCHEMBL7486775 0.85 EGFR (0.41) ALDH1A1KDM4EADORA1SMN1; SMN2MEN1
SCHEMBL5877626 0.81 ABCC1 (0.52) ALDH1A1SMN1; SMN2MEN1KMT2AABCC1
SCHEMBL5877811 0.81 ABCC1 (0.46) KMT2AABCC1AVPR1BGHSRCYP2D6
SCHEMBL5876953 0.80 ABCC1 (0.50) ALDH1A1SMN1; SMN2MEN1KMT2AABCC1
SCHEMBL5877936 0.80 CRHR1 (0.41) LMNAGHSRCYP2D6CYP3A4KCNH2
SCHEMBL6309533 0.80 ALDH1A1 (0.45) ALDH1A1KDM4ESMN1; SMN2MEN1LMNA
SCHEMBL5877732 0.80 ABCC1 (0.52) ALDH1A1MEN1KMT2AABCC1AVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed