SCHEMBL5877936

SCHEMBL5877936

COc1ccc(-c2ccc(-c3nc4ccc(C)cc4c(=O)n3CC3CCCC(CN)C3)s2)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.41
GHSR Q92847 3/20 0.38
CYP2D6 P10635 3/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
F11 P03951 1/20 0.36
P2RX3 P56373 1/20 0.36
KCNH2 Q12809 2/20 0.35
ADRA1A P35348 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP3A4 P08684 1/20 0.34
DPP4 P27487 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877056 0.96 CRHR1 (0.43) CRHR1GHSRCYP2D6GRIN1GRIN2B
SCHEMBL5877446 0.92 CRHR1 (0.41) CRHR1GHSRCYP2D6GRIN1GRIN2B
SCHEMBL5877453 0.91 CRHR1 (0.42) CRHR1GHSRLMNATP53TSHR
SCHEMBL5876985 0.89 CRHR1 (0.44) CRHR1GHSRCYP2D6GRIN1GRIN2B
SCHEMBL7488467 0.88 CRHR1 (0.41) CRHR1GHSRCYP2D6GRIN1GRIN2B
SCHEMBL5877807 0.84 F11 (0.47) CRHR1GHSRCYP2D6GRIN1GRIN2B
SCHEMBL5877943 0.83 CRHR1 (0.40) CRHR1GHSRCYP2D6GRIN1GRIN2B
SCHEMBL5877351 0.83 AVPR1B (0.40) GHSRCYP2D6F11KCNH2ADRA1A
SCHEMBL5877963 0.82 ALDH1A1 (0.47) GHSRF11KCNH2ADRA1AHRH3
SCHEMBL6313495 0.82 F11 (0.46) CRHR1F11P2RX3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed