SCHEMBL5879508

SCHEMBL5879508

NCc1csc(NC(=O)NCc2ccccc2)n1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 13/20 0.62
ROCK1 Q13464 13/20 0.62
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KCNH2 Q12809 1/20 0.51
MMP3 P08254 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3653730 0.87 ROCK2 (0.60) ROCK2ROCK1MMP3
SCHEMBL7454854 0.87 ROCK2 (0.62) ROCK2ROCK1
SCHEMBL91397 0.87 ROCK2 (0.62) ROCK2ROCK1MMP3
SCHEMBL3653731 0.86 ROCK2 (0.61) ROCK2ROCK1MMP3
Hydrochloric Acid SCHEMBL355183 0.85 ROCK1 (0.66) ROCK2ROCK1
SCHEMBL3653728 0.84 ROCK2 (0.59) ROCK2ROCK1MMP3
SCHEMBL7144846 0.83 ROCK2 (0.58) ROCK2ROCK1MMP3
SCHEMBL6316630 0.82 ROCK2 (0.62) ROCK2ROCK1MMP3
SCHEMBL6880276 0.81 ROCK2 (0.65) ROCK2ROCK1MMP3
SCHEMBL7447830 0.78 ROCK2 (0.65) ROCK2ROCK1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7125883-B1 Integrin receptor ligands ABBOTT GMBH & CO. KG (DE) 2006-10-24 US disclosed
US-7105508-B1 Integrin receptors antagonists ABBOTT GMBH & CO. KG (DE) 2006-09-12 US disclosed
US-20040259864-A1 Substituted pyrimidinone derivatives as ligands of integrin receptors ABBOTT GMBH & CO. KG (DE) 2004-12-23 US disclosed
CN-1374960-A novel integrin receptor antagonists BASF AG (DE) 2002-10-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040259864-A1 Substituted pyrimidinone derivatives as ligands of integrin receptors ITGB3, ITGA5, ITGB5 ROCK2 2519/4885ROCK1 2717/4885CYP1A2 4217/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.