SCHEMBL7454854

SCHEMBL7454854

O=C(O)Cc1csc(NC(=O)NCc2ccccc2)n1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.62
ROCK1 Q13464 3/20 0.62
ALDH1A1 P00352 1/20 0.60
SCD O00767 6/20 0.57
ITGB1 P05556 1/20 0.52
ITGA4 P13612 1/20 0.52
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51
MME P08473 1/20 0.51
PDE5A O76074 2/20 0.50
KDM4E B2RXH2 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3653730 0.90 ROCK2 (0.60) ROCK2ROCK1ALDH1A1SCDLMNA
SCHEMBL5879508 0.87 ROCK2 (0.62) ROCK2ROCK1
SCHEMBL91397 0.87 ROCK2 (0.62) ROCK2ROCK1LMNATP53
SCHEMBL3653731 0.86 ROCK2 (0.61) ROCK2ROCK1
SCHEMBL7144846 0.85 ROCK2 (0.58) ROCK2ROCK1SCDPDE5A
SCHEMBL3653728 0.84 ROCK2 (0.59) ROCK2ROCK1
SCHEMBL7016372 0.83 SCD (0.61) ALDH1A1SCDLMNAMME
SCHEMBL4781259 0.83 SCD (0.53) ROCK2ROCK1ALDH1A1SCDITGB1
SCHEMBL27743104 0.82 ALDH1A1 (0.58) ALDH1A1SCDITGB1ITGA4MME
SCHEMBL27556141 0.82 ROCK2 (0.52) ROCK2ROCK1LMNATP53PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173468-A1 INTEGRIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2002-01-23 EP disclosed
WO-2000066618-A1 INTEGRIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2000-11-09 WO disclosed