SCHEMBL5879529

SCHEMBL5879529

O=S(=O)(c1ccccc1)c1cnc2[nH]ccc(N3CCN(Cc4ccccc4)CC3)c1-2

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
DRD2 P14416 6/20 0.45
DRD4 P21917 5/20 0.45
DRD3 P35462 5/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 2/20 0.44
TRPC5 Q9UL62 1/20 0.43
HTR6 P50406 3/20 0.42
HTR2A P28223 1/20 0.41
THRB P10828 1/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5879573 0.85 HTR6 (0.52) DRD2DRD3MAPTNPSR1TDP1
SCHEMBL5879490 0.77 DRD2 (0.49) CA12CA1CA2CA9DRD2
SCHEMBL4476828 0.73 CA12 (0.52) CA12CA1CA2CA9DRD2
SCHEMBL13676941 0.72 GRM5 (0.72) MAPTL3MBTL1ALDH1A1THRB
SCHEMBL4478910 0.70 HTR6 (0.44) CA12CA1CA2CA9DRD2
SCHEMBL4494237 0.70 DRD2 (0.48) CA12CA1CA2CA9DRD2
SCHEMBL3323296 0.67 CASP1 (0.45) CA12CA1CA2CA9DRD2
SCHEMBL8242932 0.67 THRB (0.68) MAPTTDP1L3MBTL1ALDH1A1HTR6
SCHEMBL13676928 0.67 THRB (0.65) MAPTTDP1L3MBTL1ALDH1A1HTR6
SCHEMBL8238195 0.67 THRB (0.69) MAPTTDP1L3MBTL1ALDH1A1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006517966-A 2006-08-03 JP claimed
EP-1592690-A1 HETEROCYCLYL-3-SULFONYLAZAINDOLE OR -AZAINDAZOLE DERIVATIVES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2005-11-09 EP claimed
WO-2004074286-A1 HETEROCYCLYL-3-SULFONYLAZAINDOLE OR -AZAINDAZOLE DERIVATIVES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2004-09-02 WO claimed