SCHEMBL5879532

SCHEMBL5879532

CC(=O)ON1C(=O)c2ccccc2C(CC(=O)OC(C)(C)C)c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.37
BRD4 O60885 2/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
ITGB3 P05106 5/20 0.35
ITGAV P06756 5/20 0.35
CES1 P23141 1/20 0.34
TSHR P16473 1/20 0.34
PTPRC P08575 2/20 0.33
CYP1A2 P05177 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5879694 0.87 EGFR (0.41) KDRALDH1A1HPGDITGB3ITGAV
SCHEMBL5879591 0.80 ITGB3 (0.49) ITGB3ITGAV
SCHEMBL5879512 0.78 ITGB3 (0.44) HDAC3HDAC1HDAC8HDAC6ITGB3
SCHEMBL5880062 0.77 CYP1A2 (0.42) HDAC3HDAC1HDAC8HDAC6ALDH1A1
SCHEMBL5879657 0.76 EGFR (0.37) KDRALDH1A1TSHRKMT2A
SCHEMBL5879576 0.76 ITGB3 (0.54) ITGB3ITGAV
SCHEMBL5879502 0.71 ITGB3 (0.41) HDAC3HDAC1HDAC8HDAC6ITGB3
SCHEMBL7402874 0.71 BRD4 (0.39) BRD4HDAC3HDAC1HDAC8HDAC6
SCHEMBL5879521 0.69 POLB (0.46) HDAC3HDAC1HDAC8HDAC6ALDH1A1
SCHEMBL7074976 0.68 MTNR1B (0.35) HDAC3HDAC1HDAC8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7105508-B1 Integrin receptors antagonists ABBOTT GMBH & CO. KG (DE) 2006-09-12 US disclosed