SCHEMBL5887115

SCHEMBL5887115

Cc1nc(Sc2ccc(F)cc2)nc2c1ccc(=O)n2-c1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.42
MAPT P10636 1/20 0.42
RXFP1 Q9HBX9 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SMO Q99835 1/20 0.40
MAPK8 P45983 1/20 0.40
LMNA P02545 4/20 0.40
ALDH1A1 P00352 1/20 0.40
SCD O00767 1/20 0.40
HTR7 P34969 1/20 0.39
BLM P54132 1/20 0.39
AKT1 P31749 1/20 0.39
AKT2 P31751 1/20 0.39
AKT3 Q9Y243 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887077 0.91 LMNA (0.40) TP53MAPTRXFP1MAPK8LMNA
SCHEMBL5886827 0.91 PTGER4 (0.41) TP53RXFP1LMNAALDH1A1BLM
SCHEMBL5886833 0.90 CCR1 (0.43) TP53MAPTRXFP1MAPK8LMNA
SCHEMBL5887037 0.87 KLKB1 (0.41) TP53SMN1; SMN2MAPK8LMNAHTR7
SCHEMBL5886795 0.87 MAPT (0.46) TP53MAPTRXFP1MAPK8LMNA
SCHEMBL5887088 0.86 MET (0.44) TP53MAPTSMN1; SMN2ALDH1A1
SCHEMBL5886789 0.83 HPGD (0.47) TP53MAPTRXFP1SMN1; SMN2SMO
SCHEMBL5887058 0.83 TSHR (0.34) RXFP1ALDH1A1
SCHEMBL5886724 0.83 MAPT (0.41) TP53MAPTRXFP1SMN1; SMN2LMNA
SCHEMBL5886728 0.82 CTNNB1 (0.48) TP53MAPTLMNASCDHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP TP53 43/4885MAPT 1614/4885RXFP1 4707/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.